中文名稱 | 英文名稱 | CAS 號 | 用途 |
泰諾福韋系列 | |||
對甲苯磺酰氧甲基膦酸二乙酯 | Diethyl p-toluene sulfonyl oxymethyl phosphonate (DESMP) | 31618-90-3 | |
R-9-(2-磷酸氧甲基)丙基腺嘌呤 | (R)-9-[(2-Phosphonomethoxyl)propyl]Adenine (R-PMPA) | 147127-20-6 | |
(R)-(+)-9-(2-羥丙基)腺嘌呤 | (R)-9-(2-hydroxypropyl)adenine (HPA) | 14047-28-0 | |
R-碳酸丙烯酯 | R-(+)-propylene carbonate (R-PC) | 16606-55-6 | |
阿德福韋系列 | |||
9-[2-(膦酰甲氧基)乙基]腺嘌呤(阿德福韋) | 9-[2-(Phosphono Methoxy)Ethyl]Adenine (PMEA) | 106941-25-7 | |
9-[2-(二乙基膦酰甲氧基)乙基]腺嘌呤(A3) | 9-[2-(Diethyl Phosphono Methoxy)Ethyl]Adenine | 116384-53-3 | |
阿巴卡韋系列 | |||
2,5-二氨基-4,6-二羥基嘧啶鹽酸鹽 | 2,5-Diamino-4,6-dihydroxypyrimidine hydrochloride | 56830-58-1 | |
2-氨基-4,6-二氯-5-甲酰胺基嘧啶 | N-(2-Amino-4,6-dichloro-5-pyrimidinyl)formamide | 171887-03-9 | |
2-氮雜雙環[2.2.1]庚-5-烯-3-酮 | 2-Azabicyclo[2.2.1]hept-5-en-3-one (Vince lactam) | 49805-30-3 | |
度魯特韋系列 | |||
3-氨基-1-丁醇 | (R)-3-amino-1-butanol | 61477-40-5 | |
4-甲氧基乙酰乙酸甲酯 | methyl 4-methoxy-3-oxobutyrate (can be customed) | 41051-15-4 | |
阿扎那韋中間體 | |||
L-叔亮氨酸 | L-tert-leucine | 20859-02-3 | |
N-甲氧基-L-叔亮氨基酸 | N-methoxycarbonyl-L-Tert-Leucine | 162537-11-3 | |
達卡他韋系列 | |||
4,4'-二(2-溴乙?;?聯苯 | 4,4'-Bis(2-bromoacetyl)biphenyl | 4072-67-7 | |
Boc-L-脯氨酸 | Boc-L-Proline | 15761-39-4 | |
Moc-L-纈氨酸 | Moc-L-Valine | 74761-42-5 | |
地瑞那韋系列 | |||
地瑞那韋乙醇鹽 | Darunavir Ethanolate | 635728-49-3 | |
4-氨基-N-[(2R, 3S)-3-氨基-2-羥基-4-苯丁基]-N-異丁基苯磺酰胺 | 4-Amino-N-[(2r,3s)-3-Amino-2-Hydroxy-4-Phenyl butyl]-N-Isobutylbenzenesulfonamide(D7) | 169280-56-2 | |
(3AS,4S,6AR)-四氫-4-甲氧基-呋喃并[3,4-B]呋喃-2(3H)-酮 | (3aS,4S,6aR,)-4-methoxytetrahydrofuro[3,4-b]furan-2(3H)-one(SM7) | 866594-60-7 | |
(3R,3AS,6AR)-羥基六氫呋喃并[2,3-Β]呋喃基丁二酰亞胺基碳酸酯 | (3R,3aS,6aR)-Hydroxyhexahydrofuro[2,3-β]furanylSuccinimidylCarbonate(SM9) | 253265-97-3 | |
沙庫比曲系列 | |||
LCZ696中間體1 | (R)-tert-butyl (1-([1,1'-biphenyl]-4-yl)-3-hydroxypropan-2-yl)carbamate | 1426129-50-1 | |
LCZ696中間體 2 | (2R,4S)-ethyl 5-([1,1'-biphenyl]-4-yl)-4-amino-2-methylpentanoate hydrochloride | 149690-12-0 | |
LCZ696 中間體3 | 2R,4S)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)amino)-2-methylpentanoic acid | 1012341-50-2 | |
LCZ696 中間體 5 | 4-(((2S,4R)-1-([1,1'-biphenyl]-4-yl)-5-ethoxy-4-methyl-5-oxopentan-2-yl)amino)-4-oxobutanoic acid | 149709-62-6 | |
LCZ696中間體 7 | R,E)-5-([1,1'-biphenyl]-4-yl)-4-((tert-butoxycarbonyl)amino)-2-methylpent-2-enoic acid | 1012341-48-8 | |
吡啶系列 | |||
2,6-二羥基-3-氰基-4-甲基吡啶 | 2,6-Dihydroxy-3-cyano-4-methyl Pyridine | 5444-02-0 | |
2,6-二氯-3-氰基-4-甲基吡啶 | 2,6-Dichloro-3-cyano-4-methyl Pyridine | 875-35-4 | |
2,6-二氯-3-氨基-4-甲基吡啶 | 2,6-Dichloro-3-amino-4-methyl Pyridine | 129432-25-3 | |
2-氯-3-氨基-4-甲基吡啶 | 2-Chloro-3-amino-4-methyl Pyridine | 133627-45-9 | |
3-氨基-4-甲基吡啶 | 3-amino-4-methylpyriddine | 3430-27-1 | |
氟喹諾酮系列 | |||
氟氯煙腈 | 2,6-Dichloro-3-cyano-5-fluoro pyridine | 82671-02-1 | |
氟氯煙酸 | 2,6-Dichloro-5-fluoro nicotinic acid | 82671-06-5 | |
氟氯煙酯 | Ethyl 2,6-dichloro-5-fluoro nicotinoyl acetate | 96568-04-6 | |
3-(N,N-二甲基氨基)丙烯酸乙酯 | Ethyl 3-(dimethylamino)acrylate | 924-99-2 | |
莫西沙星,加替沙星中間體 | |||
加替環合酯 | 1-Cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid ethyl ester | 112811-71-9 | |
加替羧酸 | 1-Cyclopropyl-6,7-difluoro-1,4-dihydro-8-methoxy-4-oxo-3-quinolinecarboxylic acid | 112811-72-0 | |
(S,S)-2,8-二氮雜雙環[4,3,0]壬烷 | (S,S)-2,8-Diazabicyclo[4.3.0]nonane | 151213-42-2 | |
吉米沙星系列 | |||
環丙基萘啶羧酸 | 1-Cyclopropyl-6-fluoro-7-chloride-4-oxo-1,4-dihydro-1,8-naphthyridine-3-carboxylic acid | 100361-18-0 | |
環丙基萘啶羧酸乙酯 | Ethyl 1-Cyclopropyl-7-chloro-6-fluoro-1,4-dihydro-4-oxo-1,8-naphthylridine carboxylate | 96568-07-9 | |
地拉羅司系列 | |||
對肼基苯甲酸 | 4-Hydrazinobenzoic acid | 619-67-0 | |
2-(2-羥基苯基)-4H-苯并[e][1,3]惡嗪-4-酮 | 2-(2-Hydroxyphenyl)-4H-benzo[e][1,3]oxazin-4-one | 1218-69-5 | |
地拉羅司 | Deferasirox | 201530-41-8 | |
艾菲康唑系列 | |||
(2R)-1-(2,4-二氟苯基)-2-((四氫-2H-吡喃-2-基)氧)丙基-1-酮 | (2R)-1-(2,4-Difluorophenyl)-2-[(tetrahydro-2H-pyran-2-yl)oxy]-1-propanone | 126918-17-0 | |
(2R,3R)-2-(2,4-二氟苯基)-1-(1H-1,2,4-三唑-1-基)丁烷-2,3-二醇 | (2R,3R)- 2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)- 2,3-Butanediol | 133775-25-4 | |
1-(((2R,3S),2-(2,4-二氟苯基)-3-甲基環氧乙烷-2-基)甲基)-1H-1,2,4-三唑 | (2R,3S)-2-(2,4-Difluorophenyl)-3-methyl-[(1H-1,2,4-triazol-1-yl)methyl]oxirane | 127000-90-2 | |
4-亞甲基哌啶鹽酸鹽 | 4-Methylenepiperidine.HCl | 144230-50-2 | |
利拉利汀系列 | |||
1-溴-2-丁炔 | 1-Bromo-2-butyne | 3355-28-0 | |
8-溴-3-甲基黃嘌呤 | 8-Bromo-3-methyl-1H-purine-2,6-(3H,7H)-dione | 93703-24-3 | |
鄰氨基苯乙酮 | 2-Aminoacetophenone | 551-93-9 | |
2-氯甲基-4-甲基喹唑啉 | 2-Chloromethyl-4-methylquinazoline | 109113-72-6 | |
8-溴-7-(2-丁炔基)-3-甲基黃嘌呤 | 3-Methyl-7-(2-butyn-1-yl)-8-bromoxanthine | 666816-98-4 | |
8-溴-7-(2-丁炔-1-基)-3,7-二氫-3-甲基-1-[(4-甲基-2-喹唑啉基)甲基]-1H-嘌呤-2,6-二酮 | 1-[(4-methylquinazolin-2-yl)methyl]-3-methyl-7-(2-butyn-1-yl)-8-bromoxanthine | 853029-57-9 | |
(R)-3-氨基哌啶雙鹽酸鹽 | (R)-3-aminopiperidine dihydrochloride | 334618-23-4 | |
(R)-3-Boc-氨基哌啶 | (R)-3-(Boc-Amino)piperidine | 309956-78-3 | |
利拉利汀 | Linagliptin | 668270-12-0 | |
西他列汀系列 | |||
2,4,5-三氟苯乙酸 | 2,4,5-Trifluorophenyl acetic acid | 209995-38-0 | |
Boc-(R)-3-氨基-4-(2,4,5-三氟苯基)丁酸 | (R)-N-Boc-3-Amino-4-(2,4,5-trifluorophenyl) butanoic acid | 486460-00-8 | |
3-(三氟甲基)-5,6,7,8-四氫-[1,2,4]三唑并[4,3-α]吡嗪鹽酸鹽 | 3-(Trifluoromethyl)-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyrazine hydrochloride | 762240-92-6 | |
磷酸西他列汀一水合物 | Sitagliptin phosephate monohydrate | 654671-77-9 | |
維達列汀系列 | |||
3-氨基-1-金剛烷醇 | 3-Amino-1-adamantanol | 702-82-9 | |
(2S)-N-氯乙?;?2-氰基四氫吡咯 | (2S)-1-(Chloroacetyl)-2-pyrrolidinecarbonitrile | 207557-35-5 | |
維達列汀 | Vildagliptin | 274901-16-5 | |
利伐沙班系列 | |||
2-氯噻吩-5-甲酸 | 5-Chloro-2-thiophenecarboxylic acid | 24065-33-6 | |
(S)-N-縮水甘油鄰苯二甲酰亞胺 | (S)-(+)-glycidyl phthalimide | 161596-47-0 | |
4-(4-氨基苯基)嗎啡啉-3-酮 | 4-(4-aminophenyl)morpholin-3-one | 438056-69-0 | |
4-[4-[(5S)-5-(氨基甲基)-2-氧代-3-惡唑烷基]苯基]-3-嗎啉酮鹽酸鹽 | 4-[4-[(5S)-5-(Aminomethyl)-2-oxo-3-oxazolidinyl]phenyl]-3-morpholinone hydrochloride | 898543-06-1 | |
利伐沙班 | Rivaroxaban | 366789-02-8 | |
阿哌沙班 | |||
[(4-甲氧基苯基)肼基]氯乙酸乙酯 | Ethyl chloro[(4-methoxyphenyl)hydrazono]acetate | 27143-07-3 | |
5,6-二氫-3-(4-嗎啉基)-1-[4-(2-氧代-1-哌啶基)苯基]-2(1H)-吡啶酮 | 5,6-Dihydro-3-(4-morpholinyl)-1-[4-(2-oxo-1-piperidinyl)phenyl]-2(1H)-pyridinone | 545445-44-1 | |
5,6-二氫-3-(4-嗎啉基)-1-(4-硝基苯基)-2(1H)-吡啶酮 | 5,6-Dihydro-3-(4-Morpholinyl)-1-(4-Nitrophenyl)-2(1H)-Pyridinone | 503615-03-0 | |
阿哌沙班 | Apixaban | 503612-47-3 | |
依普利酮系列 | |||
依普利酮 | Eplerenone | 107724-20-9 | |
依普利酮N-1 | Eplerenone N-1 | 95716-70-4 | |
11α-羥基坎利酮 | 11ALPHA-HYDROXYCANRENONE | 192569-17-8 | |
維拉唑酮系列 | |||
5-氰基吲哚 | 5-Cyanoindole | 15861-24-2 | |
3-(4-氯代丁基)-5-氰基吲哚 | 3-(4-Chlorbutyl)-1H-indol-5-carbonitrile | 143612-79-7 | |
5-氨基苯并呋喃甲酸乙酯 | Ethyl 5-Aminobenzofuran-2-carboxylate | 174775-48-5 | |
5-(哌嗪-1-基)苯并呋喃-2-甲酰胺 | 5-(1-Piperazinyl)benzofuran-2-carboxamide | 183288-46-2 | |
阿瑞吡坦系列 | |||
(2R,3S)-2-[(1R)-1-[3,5-雙(三氟甲基)苯基]乙氧基]-3-(4-氟苯基)-嗎啉鹽酸鹽 | (2R,3S)-2-{(1R)-1-[3,5-Bis(trifluoromethyl)phenyl]ethoxy}-3-(4-fluorophenyl)morpholine hydrochloride | 171482-05-6 | |
3-氯甲基-1,2,4-三唑啉-5-酮 | 3-Chloromethyl-1,2,4-triazolin-5-one | 252742-72-6 | |
2-(2-氯-1-亞乙基)酰肼甲酸甲酯 | N-Methylcarbonyl-2-chloroacetamidrazone | 155742-64-6 | |
氯氮平系列 | |||
8-氯-5,10-二氫-11H-二苯并[b,e][1,4]二氮雜卓-11-酮 | CODD(8-chloro-11-oxo-10,11-Dihydro-5H-Dibenzo-1,4-Diazepine) | 50892-62-1 | |
替米沙坦系列 | |||
2-正丙基-4-甲基-6-(1-甲基苯并咪唑-2-基)苯并咪唑;雙咪唑 | 2-N-PROPYL-4-METHYL-6-(1-METHYL BENZIMIDAZOL-2-YL)-BENZIMIDAZOLE | 152628-02-9 | |
4'-溴甲基-2-甲酸甲酯聯苯 | Methyl 4'-bromomethyl biphenyl-2-carboxylate | 114772-38-2 | |
其它類 | |||
鳥嘌呤 (2-氨基-6-羥基嘌呤) | Guanine (2-Amino-6-hydroxypurine) | 73-40-5 | |
2,3-二氯-5,6-二氰對苯醌(DDQ) | 2,3-Dichloro-5,6-Dicyano-1,4-Benzoquinone(DDQ) | 84-58-2 | |
苯甲酰乙酸乙酯 | Ethyl Benzoylacetate | 94-02-0 | |
靛紅(98%) | Isatin(98%) | 91-56-5 | |
5-氟靛紅 | 5-Fluoro Isatin | 443-69-6 | |
N-羥乙基苯胺 | N-Hydroxyethylamine / 2-Anilinoethanol | 122-98-5 | |
3-羥基苯乙酮 | 3-Hydroxyl acetophenone | 121-71-1 | |
3-氨基-2-羥基苯乙酮 | 3-Amino-2-Hydroxyacetophenone | 70977-72-9 | |
環丙基甲酸乙酯 | Ethyl Cyclopropanecarboxylate | 4606-07-9 | |
4-硝基苯乙胺鹽酸鹽 | 4-Nitrophenethylamine hydrochloride | 29968-78-3 | |
4-(二乙氨基)水楊醛 | 4-(Diethylamino)salicylaldehyde | 17754-90-4 | |
3-氨基巴豆腈 | 3-Aminocrotononitrile | 1118-61-2 | |
3,4-二羥基苯甲醛 | 3,4-Dihydroxybenzaldehyde | 139-85-5 | |
3,3-二甲基丙烯酸 | 3,3-Dimethylacrylic acid | 541-47-9 | |
水楊酸 | Salicylic acid | 69-72-7 | |
2-噻吩乙酰氯 | 2-Thiophene acetyl chloride | 39098-97-0 | |
2-噻吩乙酸 | 2-Thiophene acetic acid | 1918-77-0 | |
磷酸吡哆醛 | Pyridoxal-5-phosphate(P5P) | 853645-22-4 | |
吡咯喹啉醌 | Pyrroloquinoline quinone(PQQ) | 72909-34-3 | |
1-氟萘 | Fluoronaphthalene | 321-38-0 | |
對羥基苯甲醛 | p-Hydroxybenzaldehyde | 123-08-0 | |
吡啶硫酮鋅 | Zinc pyrithione | 13463-41-7 | |
扁桃酸 | DL-mandelate acid | 90-64-2 |